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Home - Products - Metabolic Enzyme/Protease - PPAR - SR 16832

SR 16832

CAS No. 2088135-12-8

SR 16832( SR-16832 | SR16832 )

Catalog No. M27795 CAS No. 2088135-12-8

SR 16832 is a dual-site PPARγ inhibitor. It also inhibits the binding of endogenous ligands and transcriptional activity of PPARγ, more effectively than the orthosteric covalent antagonist GW 9662 and T 0070907.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    SR 16832
  • Note
    Research use only, not for human use.
  • Brief Description
    SR 16832 is a dual-site PPARγ inhibitor. It also inhibits the binding of endogenous ligands and transcriptional activity of PPARγ, more effectively than the orthosteric covalent antagonist GW 9662 and T 0070907.
  • Description
    SR 16832 is a dual-site PPARγ inhibitor. It also inhibits the binding of endogenous ligands and transcriptional activity of PPARγ, more effectively than the orthosteric covalent antagonist GW 9662 and T 0070907.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    SR-16832 | SR16832
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    PPAR
  • Recptor
    P2X7
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2088135-12-8
  • Formula Weight
    357.75
  • Molecular Formula
    C17H12ClN3O4
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (698.81 mM)
  • SMILES
    COc1ccc2nccc(NC(=O)c3cc(ccc3Cl)[N+]([O-])=O)c2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Stock TC, et al. Efficacy and safety of CE-224,535, an antagonist of P2X7 receptor, in treatment of patients with rheumatoid arthritis inadequately controlled by methotrexate. J Rheumatol. 2012 Apr;39(4):720-7.
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